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Table 1 Primary radioligand competitive binding assays

From: Functional characterization and analgesic effects of mixed cannabinoid receptor/T-type channel ligands

Ligand (10 μM)

Human 5-HT2A (%)

Rat 5-HT2C (%)

Rat CB1 (%)

Human CB2 (%)

NMP4

23.9

-9.3

99.3

104.4

NMP7

ND

ND

ND

ND

NMP139

7.7

-7.8

46.3

51.3

NMP140

11.2

-4.2

79.3

71.1

NMP141

11.9

-8.4

88.6

88.7

NMP144

-5.2

13

67.4

90.6

  1. ND: not determined
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Molecular Pain

ISSN: 1744-8069

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